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CYP2C19 (h), CYP2C19 (h)

Cat#: 400-0095
Species: Human
RegionRecombinant/SF9 cells
Substrate7-ethoxy-3-cyanocoumarin (CEC)
Substrate [M]2.5E-5
Km (enzyme affinity)3.5E-5 M
Vmax0.76 pmol CHC/pmol CYP1A2/min.
ReactionCEC + NADPH -> 7-hydroxy-3-cyanocoumarin (CHC) + NADP+
MethodFluorescence
Reference CompoundTranylcypromine
IC50 = 2.8 μM
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