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hERG (I[Kr]) (h)

Cat#: 100-0330
Species: Human
RegionRecombinant/CHO cells
Ligand[3H]Astemizole
Ligand [M]4E-8
Kd (binding affinity)1.0E-7
Bmax350 fmol/mg protein
Non-SpecificTerfenadine
Non-specific [M]1E-4
MethodRadioactivity
MeasurementDPM
Reference CompoundTerfenadine
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